1-(5-isoquinolinesulfonyl)-2-methylpiperazinemedical dictionary

<chemical>

A specific protein kinase c inhibitor, which inhibits superoxide release from human neutrophils stimulated with phorbol myristate acetate or synthetic diacylglycerol.

Pharmacological action: enzyme inhibitors.

Chemical name: Piperazine, 1-(5-isoquinolinylsulfonyl)-2-methyl-, (2S-(1(R*(R*)), 2alpha, 3abeta, 7abeta))-

(12 Dec 1998)